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                          Home » Products » Speciality Chemicals & Inhibitor » Bestatin

                          Bestatin

                          Bestatin
                          Bestatin
                          Product Code : 24
                          Product Description

                          CAS Number : 65391-42-6

                          Empirical Formula (Hill Notation) : C16H24N2O4 · HCl

                          Molecular Weight : 344.83

                          Beilstein Registry Number : 4628066

                          MDL number : MFCD00058004

                          PubChem Substance ID : 24278278


                          Packaging

                          1, 5 mg in glass bottle

                          10, 25 mg in poly bottle

                          100 mg in glass bottle

                          Preparation Note

                          Solubility testing in water at 25 mg/ml yields a clear solution. Stock solutions at 1 mM are expected to be stable at least one month stored at -20 °C.

                          Biochem/physiol Actions

                          A metalloprotease inhibitor selective for aminopeptidase. Bestatin is a competitive and specific inhibitor of leucine aminopeptidase, aminopeptidase B, and triamino peptidase. It inhibits aminopeptidase B at 60 nM (using arginine-β-naphthylamide as substrate) and leucine aminopeptidase at 20 nM (leucine-β-naphthylamide as substrate). It showed no inhibition of aminopeptidase A, trypsin, chymotrypsin, elastase, papain, pepsin, or themolysin. It offers promise as a novel analgesic because it protects endogenous  peptides against degradation.


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