Pristimerin

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Pristimerin

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Product Code : SRGCC80

Brand Name : S.R GROUP CHEMICALS

Price And Quantity

Minimum Order Quantity
1
Unit of Measure
Pack/Packs

Price Range
7900.00 - 60800.00 INR
Price
7900-60800 INR

Product Specifications

Boiling point
REFER C.O.A MSDS
Taste
Bitter

Molecular Weight
464.6 Kilograms (kg)
Other Names
3-hydroxy-9β,13α-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester

HS Code
3821
Melting Point
REFER C.O.A MSDS

Physical Form
Solid
Ph Level
REFER C.O.A MSDS

Structural Formula
C30H40O4
Shape
Crystal

Molecular Formula
C30H40O4
Smell
Stimulus

Shelf Life
24 Months
Density
REFER C.O.A MSDS

Usage
R&D FORMULATION
Appearance
POWDER

Classification
High Purity
Chemical Name
Other

CAS No
1258-84-0
Type
TETRA HYDROXI STEAROL

Purity(%)
98%
Color
WHITE

Product Description

DESCRIPTION

Synonyms

Celastrol methyl ester
NSC 99281

Monoacylglycerol lipase (MAGL) hydrolyzes the endogenous cannabinoid 2-arachidonoyl glycerol (2-AG), terminating its capacity to activate cannabinoid receptors. Pristimerin is a naturally occurring terpenoid that potently inhibits MAGL (IC50Â = 93 nM).1Â Its actions are rapid, reversible, and noncompetitive.1Â Pristimerin (1 Ã‚ÂµM) significantly increases 2-AG levels in isolated rat neurons, indicating that it inhibits endogenous MAGL in cultured cells.1Â Moreover, it does not increase levels of palmitoyl ethanolamide, suggesting that pristimerin does not affect the activity of fatty acid amide hydrolase (FAAH).

TECHNICAL INFORMATION

Formal Name

3-hydroxy-9ÃŽÂ²,13ÃŽÂ±-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester

CAS Number

1258-84-0

Synonyms

Celastrol methyl ester
NSC 99281

Molecular Formula

C30H40O4

Formula Weight

464.6

Purity

Ã¢Â‰Â¥98%

Formulation

A crystalline solid

SHIPPING & STORAGE

Storage

-20Ã‚Â°C

Shipping

Room temperatureÂ in continental US; may vary elsewhere

Stability

Ã¢Â‰Â¥ 2 years

Trade Information